Skip to content
Product Line: Pharmaceutical Chemicals

4-Amino-5-chloro-2,3-dihydro-7-benzofurancarboxylic acid

CAS 123654-26-2

Molecular structure of 4-Amino-5-chloro-2,3-dihydro-7-benzofurancarboxylic acid

CAS · 123654-26-2

01

Product Overview

4-Amino-5-chloro-2,3-dihydro-7-benzofurancarboxylic acid is a high-purity pharmaceutical-intermediates supplied for industrial and specialty chemical applications. Contact our team for specifications, packaging options and lead times.

02

Product Specifications

Appearance: Off-white to light brown (Solid)
1 H NMR Spectrum: Consistent with structure
Purity(HPLC): 98.0% min
03

Applications

 

 

1. Pharmaceutical Intermediate

This compound serves as an intermediate in the synthesis of pharmaceutical agents, especially antibacterial or anti-inflammatory drugs.

Benzofuran derivatives are known scaffolds in medicinal chemistry for their biological activity.

2. Building Block in Organic Synthesis

Due to the presence of functional groups (amino, chloro, and carboxylic acid), this compound is versatile for:

Amide coupling reactions

Substitution reactions at the chloro position

Heterocyclic synthesis or derivatization

3. Research and Development

Used in academic and industrial R&D for designing novel small molecules or drug candidates.

4. Agrochemical Development

Potential intermediate in the synthesis of herbicides or plant growth regulators, owing to its benzofuran backbone.

04

Benefits

Multifunctional Reactivity: Its three reactive groups allow broad synthetic modification options.

Biological Potential: As a benzofuran derivative, it holds promise for pharmacological profiling.

Custom Derivatization: Useful in SAR (Structure-Activity Relationship) studies by modifying one or more functional sites.

Synthetic Flexibility: The molecule can undergo numerous transformations, such as esterification, amidation, or halogen exchange.

05

Conclusion

4-Amino-5-chloro-2,3-dihydro-7-benzofurancarboxylic acid (CAS 123654-26-2) is a valuable compound in the field of pharmaceutical and chemical synthesis. Its multifunctional nature and biologically active core structure make it a suitable intermediate for drug discovery, agrochemical development, and advanced organic chemistry. With its versatile reactivity, it supports innovation in synthesizing novel functional molecules.

Previous

Methyl Alpha-D-galactopyranoside丨CAS 3396-99-4

Next

Diethyl 5-amino-3-methylthiophene-2,4-dicarboxylate丨CAS 4815-30-9