Skip to content
Product Line: Pharmaceutical Chemicals

(1S)-4,5-Dimethoxy-1-[(methylamino)methyl]benzocyclobutane hydrochloride

CAS 866783-13-3

Molecular structure of (1S)-4,5-Dimethoxy-1-[(methylamino)methyl]benzocyclobutane hydrochloride

CAS · 866783-13-3

01

Product Overview

(1S)-4,5-Dimethoxy-1-[(methylamino)methyl]benzocyclobutane hydrochloride is a high-purity pharmaceutical-intermediates supplied for industrial and specialty chemical applications. Contact our team for specifications, packaging options and lead times.

02

Product Specifications

Appearance White or off-white powder
Assay 98.0% min
Identification (HPLC) Retention time of the sample conforms to that of the reference standard
Related substances (%Area Normalization, By HPLC) Any single impurity: 0.50% max Total impurities: 2.0% max Purity: 98.0% min
Water 1.0% max
Isomer 0.5% max
Loss on drying 1.0% max
03

Applications

(1S)-4,5-Dimethoxy-1-[(methylamino)methyl]benzocyclobutane hydrochloride is primarily used as a synthetic intermediate in pharmaceutical and medicinal chemistry. It serves as a building block for the development of central nervous system (CNS) active compounds, including neuroactive agents and psychoactive research chemicals. The compound is utilized in the synthesis of analogs for studying neurotransmitter pathways, receptor binding, and CNS-related pharmacological effects. It is also applied in research focused on drug discovery and optimization of biologically active small molecules.

04

Benefits

The benefits of this compound include its well-defined stereochemistry and functional groups, which allow for selective reactions and efficient incorporation into complex molecular structures. Its hydrochloride form enhances stability and solubility, making it easier to handle in laboratory and synthetic procedures. By providing a versatile scaffold, it supports the design of molecules with specific pharmacological profiles, facilitating studies in neurochemistry, receptor modulation, and therapeutic development. Its structural properties contribute to predictable reactivity and high yield in multi-step synthesis.

05

Conclusion

(1S)-4,5-Dimethoxy-1-[(methylamino)methyl]benzocyclobutane hydrochloride is a valuable intermediate for CNS-related pharmaceutical research and drug development. Its stereochemical precision, functional versatility, and stability make it essential for constructing complex bioactive molecules. By enabling targeted synthesis and facilitating exploration of neuroactive compounds, it continues to play a key role in medicinal chemistry and pharmacological studies.

Previous

Tosyl Isocyanate丨CAS 4083-64-1

Next

3-Chloroperoxybenzoic Acid丨CAS 937-14-4