CAS · 136310-64-0
Product Overview
Scopine-2,2-dithienyl glycolate is a high-purity pharmaceutical-intermediates supplied for industrial and specialty chemical applications. Contact our team for specifications, packaging options and lead times.
Product Specifications
| Appearance | Off-white to light pink little crystal powder |
|---|---|
| Solubility | Solubility in methylene dichloride |
| Purity | 99% min |
| Isomer | 0.1% max |
| Related substance | |
| Single impurity | 0.3% max |
| Total impurity | 1.0% max |
| Melting point | 145~153 °C |
Applications
Scopine-2,2-dithienyl glycolate is mainly used as a pharmaceutical intermediate in medicinal chemistry and drug development. It is a key structural component in the synthesis of antimuscarinic and anticholinergic agents, where the scopine moiety contributes to receptor binding and biological activity. The compound is applied in research focused on central nervous system and respiratory indications, supporting the development of therapeutics that target muscarinic acetylcholine receptors. In laboratory settings, it is also used for structure–activity relationship studies, optimization of ester-linked tropane derivatives, and exploration of pharmacological profiles of substituted glycolate esters.
Benefits
The compound offers several advantages due to its unique combination of a rigid scopine framework and a lipophilic dithienyl glycolate group. This structural arrangement enhances receptor affinity and selectivity in target molecules, supporting improved pharmacological performance. The ester linkage allows controlled chemical modification and hydrolysis, providing flexibility during synthesis and optimization. Its well-defined stereochemistry ensures predictable biological and chemical behavior, reducing variability in research outcomes. Additionally, the compound is compatible with standard organic synthesis techniques and solvents, facilitating efficient incorporation into multi-step pharmaceutical synthesis processes.
Conclusion
Scopine-2,2-dithienyl glycolate is a valuable intermediate for pharmaceutical research and drug development. Its applications in the synthesis of antimuscarinic agents, combined with benefits such as structural rigidity, chemical versatility, and reproducible performance, make it an important compound for advancing medicinal chemistry programs and the development of therapeutically relevant molecules.
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